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Catalogue
Number
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Product
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Order number / Unit
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2056
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Buprenorphin hydrochloride
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2056.0030: 30 mg per vial
Please inquire for customized
filling and bulk quantities.
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Reference standard for 6-O-[11C]-buprenorphine
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Controlled substance, license required in most countries.
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Molar Mass: 504.10
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C29H41NO4 ⋅ HCl
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[53152-21-9]
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Colourless to off-white crystalline powder packaged in dark glass crimp cap vials.
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Purity: > 95 %
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Certificates:
CoA; 1H and 13C NMR spectra
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Chemical Name:
CA index names: 6,14-Ethenomorphinan-7-methanol, 17-(cyclopropylmethyl)-α-(1,1-dimethylethyl)-4,5-epoxy-18,19-dihydro-3-hydroxy-6-methoxy-α-methyl-, hydrochloride (1:1); 6,14-Ethenomorphinan-7-methanol, 17-(cyclopropylmethyl)-α-(1,1-dimethylethyl)-4,5-epoxy-18,19-dihydro-3-hydroxy-6-methoxy-α-methyl-, hydrochloride, [5α,7α(S)]-; 6,14-Ethenomorphinan-7-methanol, 17-(cyclopropylmethyl)-α-(1,1-dimethylethyl)-4,5-epoxy-18,19-dihydro-3-hydroxy-6-methoxy-α-methyl-, hydrochloride, (αS,5α,7α)-
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Synonymes:
Buprederm; Buprenex; Buprenorphine hydrochloride
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Literature:
1. Luthra S. K. et al.: Automated radiosynthesis of [6-O-methyl-11C]-diprenorphine and [6-O-methyl-11C]-buprenorphine from 3-O-trityl protected precursors. Appl. Radiat. Isot. 1994, 45, 857-887.
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2. Luthra S.K. et al. Preparation of [11C]buprenorphine - A potential radioligand for the study of the opiate receptor system in vivo. Int. J. Rad. Appl. Instrum. A. 1987, 38, 65-6.
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3. Lever J.R. et al. Facile synthesis of [11C]buprenorphine for positron emission tomographic studies of opioid receptors. J. Rad. Appl. Instrum. A, 1990, 41, 745-52.
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4. Shiue C.Y. et al. A comparison of the brain uptake of N-(cyclopropyl[11C]methyl)norbuprenorphine ([11C]buprenorphine) and N-(cyclopropyl[11C]methyl)nordiprenorphine ([11C]diprenorphine) in baboon using PET. Int. J. Rad. Appl. Instrum. B. 1991, 18, 281-8.
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date of product catalogue issue:
05 April 2012
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